The site has moved. Please update your bookmarks.

If you are not redirected, click here to access the PDSP IMS site.




The database has 60243Ki values for searching, and is growing
This list shows the Top 100 Receptors/Targets in Ki
Please let us know if you feel we should add any papers or data. We welcome all feedback/suggestions/comments
Other features on Ki DB are: Download Ki, Data Mining, CDD Interface allows mining Ki database by structure, substructure or structure similarity.
Anatomical profiling of GPCR expression is offered for selected targets.

Make a new search

Your search returned 10 results:

IDReceptor/AliasesUniGeneAnat. ProfilingTest Ligand Name/AliasesNCIKi (nM)PubChemChEMBLHot Ligand/AliasesSpeciesSourceReference
1737 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling CHLORPHENIRAMINE  Aliases N/A 2,980.470000 PubChem-Compound ChEMBL 125I-MIL  Aliases RAT CORTEX HOFFMAN ET AL., 1987
 
902 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling CHLORPHENIRAMINE  Aliases N/A 5,000.000000 PubChem-Compound ChEMBL 125I-LSD  Aliases MOUSE C. PLEXUS TUM YAGALOFF ET AL., 1986
 
901 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling CHLORPHENIRAMINE  Aliases N/A 3,120.000000 PubChem-Compound ChEMBL 3H-MIANSERIN  Aliases RAT Choroid Plexus Sanders-Bush E, Breeding M., 1988
 
11037 HISTAMINE H1  Aliases NCBI - UniGene Anatomical Profiling CHLORPHENIRAMINE  Aliases N/A 2.510000 PubChem-Compound ChEMBL 3H-MEPYRAMINE  Aliases HUMAN CLONED Moguilevsky N et al, 1994
11906 HISTAMINE H1  Aliases NCBI - UniGene Anatomical Profiling CHLORPHENIRAMINE  Aliases N/A 2.510000 PubChem-Compound ChEMBL 3H-MEPYRAMINE  Aliases HUMAN CLONED Moguilevsky N, et al., 1995
Average2.51 
11952 HISTAMINE H1  Aliases NCBI - UniGene Anatomical Profiling CHLORPHENIRAMINE  Aliases N/A 3.000000 PubChem-Compound ChEMBL 3H-MEPYRAMINE  Aliases HUMAN FR. CORTEX Arias-Montano, et al., 1993
 
11045 HISTAMINE H1  Aliases NCBI - UniGene Anatomical Profiling CHLORPHENIRAMINE  Aliases N/A 0.500000 PubChem-Compound ChEMBL 3H-MEPYRAMINE  Aliases GUINEA PIG CEREBELLUM Moguilevsky N et al, 1994
 
9600 HISTAMINE H1  Aliases NCBI - UniGene Anatomical Profiling CHLORPHENIRAMINE  Aliases N/A 0.440000 PubChem-Compound ChEMBL 3H-PYRILAMINE  Aliases GUINEA PIG BRAIN Owens MJ, et al, 1997
 
11729 HISTAMINE H3  Aliases NCBI - UniGene Anatomical Profiling CHLORPHENIRAMINE  Aliases N/A > 10,000.000000 PubChem-Compound ChEMBL 3H-RAMHA  Aliases RAT BRAIN West RE Jr., et al., 1990
 
14430 HISTAMINE H4  Aliases NCBI - UniGene N/A CHLORPHENIRAMINE  Aliases N/A 2,910.000000 PubChem-Compound ChEMBL 3H-PYRILAMINE  Aliases HUMAN CLONED Nguyen T. et al., 2001
 


Ki ID:  
Receptor:
Receptor:
Species:
Species:
Source:
Source:
Hot Ligand:
Hot Ligand:
Test Ligand:
Test Ligand:
Reference: