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The database has 60243Ki values for searching, and is growing
This list shows the Top 100 Receptors/Targets in Ki
Please let us know if you feel we should add any papers or data. We welcome all feedback/suggestions/comments
Other features on Ki DB are: Download Ki, Data Mining, CDD Interface allows mining Ki database by structure, substructure or structure similarity.
Anatomical profiling of GPCR expression is offered for selected targets.

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Your search returned 14 results:

IDReceptor/AliasesUniGeneAnat. ProfilingTest Ligand Name/AliasesNCIKi (nM)PubChemChEMBLHot Ligand/AliasesSpeciesSourceReference
45595 5-HT Transporter  Aliases NCBI - UniGene N/A IPRINDOLE  Aliases 169449 1,620.000000 PubChem-Compound ChEMBL 3H-IMIPRAMINE  Aliases HUMAN CLONED Tatsumi M, et al., 1997
 
4472 5-HT Transporter  Aliases NCBI - UniGene N/A IPRINDOLE  Aliases 169449 1,000.000000 PubChem-Compound ChEMBL 3H-IMIPRAMINE  Aliases RAT BRAIN PALVIMAKI EP, ET AL., 1996
 
4455 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling IPRINDOLE  Aliases 169449 217.000000 PubChem-Compound ChEMBL 3H-KETANSERIN  Aliases RAT CLONED PALVIMAKI EP, ET AL., 1996
 
4437 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling IPRINDOLE  Aliases 169449 206.000000 PubChem-Compound ChEMBL 3H-MESULERGINE  Aliases RAT CLONED PALVIMAKI EP, ET AL., 1996
 
13307 adrenergic Beta  Aliases NCBI - UniGene Anatomical Profiling IPRINDOLE  Aliases 169449 > 10,000.000000 PubChem-Compound ChEMBL 3H-DHA  Aliases Mammalian BRAIN Bylund DB, et al., 1976
 
62821 Alpha 1 Adrenergic Receptor  Aliases N/A N/A IPRINDOLE  Aliases 169449 2,300.000000 PubChem-Compound ChEMBL 3H-PRAZOSIN  Aliases HUMAN Brain Frontal Cortex Richelson, Elliott et. al, 1984
 
62845 Alpha 2 Adrenergic Receptor  Aliases N/A N/A IPRINDOLE  Aliases 169449 8,600.000000 PubChem-Compound ChEMBL 3H-RAUWOLSCINE  Aliases HUMAN Brain Frontal Cortex Richelson, Elliott et. al, 1984
 
45597 Dopamine Transporter  Aliases NCBI - UniGene N/A IPRINDOLE  Aliases 169449 6,530.000000 PubChem-Compound ChEMBL 3H-WIN 35,428  Aliases HUMAN CLONED Tatsumi M, et al., 1997
 
62763 H1  Aliases N/A N/A IPRINDOLE  Aliases 169449 130.000000 PubChem-Compound ChEMBL 3H-doxepin  Aliases HUMAN Brain Frontal Cortex Richelson, Elliott et. al, 1984
 
12009 HISTAMINE H1  Aliases NCBI - UniGene Anatomical Profiling IPRINDOLE  Aliases 169449 120.000000 PubChem-Compound ChEMBL 3H-doxepin  Aliases HUMAN CORTICAL MEMBRANES Kanba S, et al., 1984
 
13057 HISTAMINE H1  Aliases NCBI - UniGene Anatomical Profiling IPRINDOLE  Aliases 169449 100.000000 PubChem-Compound ChEMBL 3H-MEPYRAMINE  Aliases RAT BRAIN Tran VT, et al., 1978
 
62789 Muscarinic Acetylcholine Receptor  Aliases N/A N/A IPRINDOLE  Aliases 169449 2,100.000000 PubChem-Compound ChEMBL 3H-QNB  Aliases HUMAN Brain caudate nucleus Richelson, Elliott et. al, 1984
 
45596 Norepinephrine transporter  Aliases N/A N/A IPRINDOLE  Aliases 169449 1,262.000000 PubChem-Compound ChEMBL 3H-Nisoxetine  Aliases HUMAN CLONED Tatsumi M, et al., 1997
 
47553 Sigma  Aliases N/A N/A IPRINDOLE  Aliases 169449 > 10,000.000000 PubChem-Compound ChEMBL 3H-3-PPP,(+)  Aliases RAT BRAIN Largent BL, et al., 1984
 


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