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The database has 60243Ki values for searching, and is growing
This list shows the Top 100 Receptors/Targets in Ki
Please let us know if you feel we should add any papers or data. We welcome all feedback/suggestions/comments
Other features on Ki DB are: Download Ki, Data Mining, CDD Interface allows mining Ki database by structure, substructure or structure similarity.
Anatomical profiling of GPCR expression is offered for selected targets.

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Your search returned 57 results:

IDReceptor/AliasesUniGeneAnat. ProfilingTest Ligand Name/AliasesNCIKi (nM)PubChemChEMBLHot Ligand/AliasesSpeciesSourceReference
41653 5-HT Transporter  Aliases NCBI - UniGene N/A N-DESMETHYLCLOZAPINE  Aliases N/A 316.600000 PubChem-Compound N/A 3H-CITALOPRAM  Aliases HUMAN CLONED PDSP certified data
 
41610 5-HT1A  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 13.900000 PubChem-Compound N/A 3H-8-OH-DPAT  Aliases HUMAN CLONED PDSP certified data
 
41611 5-HT1B  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 406.800000 PubChem-Compound N/A 3H-GR-125743  Aliases HUMAN CLONED PDSP certified data
 
41612 5-HT1D  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 476.200000 PubChem-Compound N/A 3H-GR-125743  Aliases HUMAN CLONED PDSP certified data
 
41613 5-HT1E  Aliases NCBI - UniGene N/A N-DESMETHYLCLOZAPINE  Aliases N/A 393.400000 PubChem-Compound N/A 3H-5HT  Aliases HUMAN CLONED PDSP certified data
 
41614 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 10.900000 PubChem-Compound N/A 3H-KETANSERIN  Aliases HUMAN CLONED PDSP certified data
 
41620 5-HT2B  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 2.800000 PubChem-Compound N/A 3H-LSD  Aliases HUMAN CLONED PDSP certified data
 
41615 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 11.900000 PubChem-Compound N/A 3H-MESULERGINE  Aliases RAT CLONED PDSP certified data
 
41616 5-HT3  Aliases NCBI - UniGene N/A N-DESMETHYLCLOZAPINE  Aliases N/A 272.200000 PubChem-Compound N/A 3H-ZACOPRIDE  Aliases HUMAN CLONED PDSP certified data
 
41617 5-HT5  Aliases N/A N/A N-DESMETHYLCLOZAPINE  Aliases N/A 350.600000 PubChem-Compound N/A 3H-LSD  Aliases HUMAN CLONED PDSP certified data
 
41618 5-HT6  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 11.600000 PubChem-Compound N/A 3H-LSD  Aliases HUMAN CLONED PDSP certified data
 
3129 5-HT6  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 9.400000 PubChem-Compound N/A 3H-LSD  Aliases RAT CLONED ROTH ET AL., 1993
 
41619 5-HT7  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 60.100000 PubChem-Compound N/A 3H-LSD  Aliases HUMAN CLONED PDSP certified data
 
3169 5-HT7  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 14.900000 PubChem-Compound N/A 3H-LSD  Aliases RAT CLONED ROTH ET AL., 1993
 
41621 adrenergic Alpha1A  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 104.800000 PubChem-Compound N/A 3H-PRAZOSIN  Aliases HUMAN CLONED PDSP certified data
 
41622 adrenergic Alpha1B  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 85.200000 PubChem-Compound N/A 3H-PRAZOSIN  Aliases HUMAN CLONED PDSP certified data
 
41623 adrenergic Alpha2A  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 137.600000 PubChem-Compound N/A 3H-CLONIDINE  Aliases HUMAN CLONED PDSP certified data
 
41624 adrenergic Alpha2B  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 95.100000 PubChem-Compound N/A 3H-CLONIDINE  Aliases HUMAN CLONED PDSP certified data
 
41625 adrenergic Alpha2C  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 117.700000 PubChem-Compound N/A 3H-CLONIDINE  Aliases HUMAN CLONED PDSP certified data
 
41626 adrenergic Beta1  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 6,239.040000 PubChem-Compound N/A 125I-Pindolol  Aliases HUMAN CLONED PDSP certified data
 
41627 adrenergic Beta2  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 4,725.000000 PubChem-Compound N/A 125I-Pindolol  Aliases HUMAN CLONED PDSP certified data
 
41645 Calcium channel  Aliases N/A N/A N-DESMETHYLCLOZAPINE  Aliases N/A > 10,000.000000 PubChem-Compound N/A 3H-Nitrendipine  Aliases RAT HEART PDSP certified data
 
41646 CANNABINOID CB1  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A > 10,000.000000 PubChem-Compound N/A 3H-CP-55940  Aliases RAT BRAIN PDSP certified data
 
41647 CANNABINOID CB2  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A > 10,000.000000 PubChem-Compound N/A 3H-CP-55940  Aliases HUMAN CLONED PDSP certified data
 
41639 Cholinergic, muscarinic M1  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 67.600000 PubChem-Compound N/A 3H-QNB  Aliases HUMAN CLONED PDSP certified data
 
41640 Cholinergic, muscarinic M2  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 414.500000 PubChem-Compound N/A 3H-QNB  Aliases HUMAN CLONED PDSP certified data
 
41641 Cholinergic, muscarinic M3  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 95.700000 PubChem-Compound N/A 3H-QNB  Aliases HUMAN CLONED PDSP certified data
 
41642 Cholinergic, muscarinic M4  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 169.900000 PubChem-Compound N/A 3H-QNB  Aliases HUMAN CLONED PDSP certified data
 
41643 Cholinergic, muscarinic M5  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 35.400000 PubChem-Compound N/A 3H-QNB  Aliases HUMAN CLONED PDSP certified data
 
41632 DOPAMINE D1  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 14.300000 PubChem-Compound N/A 3H-SCH23390  Aliases HUMAN CLONED PDSP certified data
 
41633 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 115.200000 PubChem-Compound N/A 3H-NMSP  Aliases HUMAN CLONED PDSP certified data
 
39073 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 89.000000 PubChem-Compound N/A R-SAT  Aliases HUMAN CLONED Burstein ES, et al., 2005
 
19742 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 100.000000 PubChem-Compound N/A UNDEFINED  Aliases HUMAN CLONED Seeman P, Tallerico T., 1998
 
41634 DOPAMINE D3  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 234.000000 PubChem-Compound N/A 3H-NMSP  Aliases RAT CLONED PDSP certified data
 
39143 DOPAMINE D3  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 153.000000 PubChem-Compound N/A R-SAT  Aliases HUMAN CLONED Burstein ES, et al., 2005
 
41635 DOPAMINE D4  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 101.820000 PubChem-Compound N/A 3H-NMSP  Aliases HUMAN CLONED PDSP certified data
 
39175 DOPAMINE D4  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 70.000000 PubChem-Compound N/A R-SAT  Aliases HUMAN CLONED Burstein ES, et al., 2005
 
19819 DOPAMINE D4  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 20.000000 PubChem-Compound N/A UNDEFINED  Aliases HUMAN CLONED Seeman P, Tallerico T., 1998
 
41636 DOPAMINE D5  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 283.600000 PubChem-Compound N/A 3H-SCH23390  Aliases HUMAN CLONED PDSP certified data
 
41637 Dopamine Transporter  Aliases NCBI - UniGene N/A N-DESMETHYLCLOZAPINE  Aliases N/A > 10,000.000000 PubChem-Compound N/A 3H-WIN 35,428  Aliases HUMAN CLONED PDSP certified data
 
41649 GABA A  Aliases N/A N/A N-DESMETHYLCLOZAPINE  Aliases N/A > 10,000.000000 PubChem-Compound N/A 3H-MUSCIMOL  Aliases RAT FOREBRAIN PDSP certified data
 
41652 Glutamate-NMDA-MK801  Aliases N/A N/A N-DESMETHYLCLOZAPINE  Aliases N/A > 10,000.000000 PubChem-Compound N/A 3H-MK-801  Aliases RAT FOREBRAIN PDSP certified data
 
41628 HISTAMINE H1  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 3.400000 PubChem-Compound N/A 3H-PYRILAMINE  Aliases HUMAN CLONED PDSP certified data
 
41629 HISTAMINE H2  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 345.100000 PubChem-Compound N/A 3H-TIOTIDINE  Aliases HUMAN CLONED PDSP certified data
 
41630 HISTAMINE H3  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A > 10,000.000000 PubChem-Compound N/A 3H-Alpha-Me-histamine  Aliases GUINEA PIG CLONED PDSP certified data
 
41631 HISTAMINE H4  Aliases NCBI - UniGene N/A N-DESMETHYLCLOZAPINE  Aliases N/A 1,028.000000 PubChem-Compound N/A 3H-Histamine  Aliases HUMAN CLONED PDSP certified data
 
41650 Imidazoline I1  Aliases N/A N/A N-DESMETHYLCLOZAPINE  Aliases N/A 757.300000 PubChem-Compound N/A 125I-Pindolol  Aliases RAT PC12 PDSP certified data
 
41638 Norepinephrine transporter  Aliases N/A N/A N-DESMETHYLCLOZAPINE  Aliases N/A 493.900000 PubChem-Compound N/A 3H-Nisoxetine  Aliases HUMAN CLONED PDSP certified data
 
41608 OPIATE Delta  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A 127.900000 PubChem-Compound N/A 3H-DADLE  Aliases HUMAN CLONED PDSP certified data
 
41609 OPIATE Kappa  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A > 10,000.000000 PubChem-Compound N/A 3H-Diprenorphine  Aliases HUMAN CLONED PDSP certified data
 
41651 OPIATE Mu  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A > 10,000.000000 PubChem-Compound N/A 3H-Diprenorphine  Aliases HUMAN CLONED PDSP certified data
 
41648 Prostaglandin E3  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A > 10,000.000000 PubChem-Compound N/A 3H-PGE2  Aliases HUMAN CLONED PDSP certified data
 
41654 Sigma-1  Aliases N/A N/A N-DESMETHYLCLOZAPINE  Aliases N/A > 10,000.000000 PubChem-Compound N/A 3H-Pentazocine(+)  Aliases RAT BRAIN PDSP certified data
 
41656 Sigma-2  Aliases N/A N/A N-DESMETHYLCLOZAPINE  Aliases N/A > 10,000.000000 PubChem-Compound N/A 3H-DTG  Aliases RAT PC12 PDSP certified data
 
41655 VASOPRESSIN V1  Aliases N/A N/A N-DESMETHYLCLOZAPINE  Aliases N/A > 10,000.000000 PubChem-Compound N/A 3H-VASOPRESSIN  Aliases HUMAN CLONED PDSP certified data
 
41658 VASOPRESSIN V2  Aliases NCBI - UniGene Anatomical Profiling N-DESMETHYLCLOZAPINE  Aliases N/A > 10,000.000000 PubChem-Compound N/A 3H-VASOPRESSIN  Aliases HUMAN CLONED PDSP certified data
 
41657 Vasopressin V3  Aliases N/A N/A N-DESMETHYLCLOZAPINE  Aliases N/A > 10,000.000000 PubChem-Compound N/A 3H-VASOPRESSIN  Aliases HUMAN CLONED PDSP certified data
 


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