The site has moved. Please update your bookmarks.

If you are not redirected, click here to access the PDSP IMS site.




The database has 60243Ki values for searching, and is growing
This list shows the Top 100 Receptors/Targets in Ki
Please let us know if you feel we should add any papers or data. We welcome all feedback/suggestions/comments
Other features on Ki DB are: Download Ki, Data Mining, CDD Interface allows mining Ki database by structure, substructure or structure similarity.
Anatomical profiling of GPCR expression is offered for selected targets.

Make a new search

Your search returned 20 results:

IDReceptor/AliasesUniGeneAnat. ProfilingTest Ligand Name/AliasesNCIKi (nM)PubChemChEMBLHot Ligand/AliasesSpeciesSourceReference
34471 5-HT Transporter  Aliases NCBI - UniGene N/A BUPRENORPHINE  Aliases N/A > 10,000.000000 PubChem-Compound N/A 3H-5HT  Aliases RAT CEREBRAL CORTEX Codd EE et al, 1995
 
34446 Norepinephrine transporter  Aliases N/A N/A BUPRENORPHINE  Aliases N/A > 10,000.000000 PubChem-Compound N/A 3H-Norepinephrine  Aliases RAT medulla, pons Codd EE et al, 1995
 
34394 OPIATE Delta  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 25.800000 PubChem-Compound N/A 3H-DPDPE  Aliases RAT FOREBRAIN Codd EE et al, 1995
 
10943 OPIATE Delta  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 1.300000 PubChem-Compound N/A 3H-DPDPE  Aliases GUINEA PIG BRAIN TRAYNOR, JR., et al., 1999
 
3711 OPIATE Delta  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 4.500000 PubChem-Compound N/A 3H-DPDPE-Cl  Aliases HUMAN CLONED TOLL L, et. al., 1998
 
3712 OPIATE Delta  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 1.600000 PubChem-Compound N/A 3H-DPDPE-Cl  Aliases GUINEA PIG BRAIN TOLL L, et. al., 1998
 
51988 OPIATE Delta  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 4.500000 PubChem-Compound N/A UNDEFINED  Aliases HUMAN UNDEFINED Rennison D et al., 2007
55918 OPIATE Delta  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 2.900000 PubChem-Compound N/A UNDEFINED  Aliases HUMAN UNDEFINED Wentland MP et al., 2009
Average3.70 
10949 OPIATE Kappa  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 2.000000 PubChem-Compound N/A 3H-CI977  Aliases GUINEA PIG BRAIN TRAYNOR, JR., et al., 1999
 
3713 OPIATE Kappa  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 0.800000 PubChem-Compound N/A 3H-U69,593  Aliases HUMAN CLONED TOLL L, et. al., 1998
 
34420 OPIATE Kappa  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 12.900000 PubChem-Compound N/A 3H-U69,593  Aliases RAT FOREBRAIN Codd EE et al, 1995
 
3714 OPIATE Kappa  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 1.500000 PubChem-Compound N/A 3H-U69,593  Aliases GUINEA PIG BRAIN TOLL L, et. al., 1998
 
51963 OPIATE Kappa  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 0.800000 PubChem-Compound N/A UNDEFINED  Aliases HUMAN UNDEFINED Rennison D et al., 2007
55947 OPIATE Kappa  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 0.620000 PubChem-Compound N/A UNDEFINED  Aliases HUMAN UNDEFINED Wentland MP et al., 2009
Average0.71 
3405 OPIATE Mu  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 1.500000 PubChem-Compound N/A 3H-DAMGO  Aliases HUMAN CLONED TOLL L, et. al., 1998
 
34368 OPIATE Mu  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 4.180000 PubChem-Compound N/A 3H-DAMGO  Aliases RAT FOREBRAIN Codd EE et al, 1995
 
3710 OPIATE Mu  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 1.300000 PubChem-Compound N/A 3H-DAMGO  Aliases GUINEA PIG BRAIN TOLL L, et. al., 1998
10937 OPIATE Mu  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 0.570000 PubChem-Compound N/A 3H-DAMGO  Aliases GUINEA PIG BRAIN TRAYNOR, JR., et al., 1999
Average0.94 
51938 OPIATE Mu  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 1.500000 PubChem-Compound N/A UNDEFINED  Aliases HUMAN UNDEFINED Rennison D et al., 2007
55889 OPIATE Mu  Aliases NCBI - UniGene Anatomical Profiling BUPRENORPHINE  Aliases N/A 0.210000 PubChem-Compound N/A UNDEFINED  Aliases HUMAN UNDEFINED Wentland MP et al., 2009
Average0.85 


Ki ID:  
Receptor:
Receptor:
Species:
Species:
Source:
Source:
Hot Ligand:
Hot Ligand:
Test Ligand:
Test Ligand:
Reference: