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The database has 60243Ki values for searching, and is growing
This list shows the Top 100 Receptors/Targets in Ki
Please let us know if you feel we should add any papers or data. We welcome all feedback/suggestions/comments
Other features on Ki DB are: Download Ki, Data Mining, CDD Interface allows mining Ki database by structure, substructure or structure similarity.
Anatomical profiling of GPCR expression is offered for selected targets.

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Your search returned 19 results:

IDReceptor/AliasesUniGeneAnat. ProfilingTest Ligand Name/AliasesNCIKi (nM)PubChemChEMBLHot Ligand/AliasesSpeciesSourceReference
37196 5-HT Transporter  Aliases NCBI - UniGene N/A Dothiepin  Aliases 172130 78.000000 PubChem-Compound N/A 3H-5-HT Uptake  Aliases RAT BRAIN Sanchez C, et al., 1999
 
47712 5-HT Transporter  Aliases NCBI - UniGene N/A Dothiepin  Aliases 172130 77.800000 PubChem-Compound N/A 3H-5-HT Uptake  Aliases RAT FR. CORTEX Cheetham SC, et.al., 1993
 
45574 5-HT Transporter  Aliases NCBI - UniGene N/A Dothiepin  Aliases 172130 8.600000 PubChem-Compound N/A 3H-IMIPRAMINE  Aliases HUMAN CLONED Tatsumi M, et al., 1997
 
47690 5-HT Transporter  Aliases NCBI - UniGene N/A Dothiepin  Aliases 172130 31.300000 PubChem-Compound N/A 3H-PAROXETINE  Aliases RAT FR. CORTEX Cheetham SC, et.al., 1993
 
37229 5-HT1A  Aliases NCBI - UniGene Anatomical Profiling Dothiepin  Aliases 172130 4,004.000000 PubChem-Compound N/A 3H-8-OH-DPAT  Aliases RAT CORTEX Sanchez C, et al., 1999
 
37240 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling Dothiepin  Aliases 172130 152.000000 PubChem-Compound N/A 3H-KETANSERIN  Aliases RAT CORTEX Sanchez C, et al., 1999
 
37279 adrenergic Alpha1  Aliases N/A N/A Dothiepin  Aliases 172130 419.000000 PubChem-Compound N/A 3H-PRAZOSIN  Aliases RAT CORTEX Sanchez C, et al., 1999
 
37290 adrenergic Alpha2  Aliases N/A N/A Dothiepin  Aliases 172130 12.000000 PubChem-Compound N/A 3H-IDAZOXAN  Aliases RAT CORTEX Sanchez C, et al., 1999
 
37310 Cholinergic, muscarinic  Aliases N/A N/A Dothiepin  Aliases 172130 26.000000 PubChem-Compound N/A 3H-QNB  Aliases RAT BRAIN Sanchez C, et al., 1999
 
41991 Cholinergic, muscarinic M1  Aliases NCBI - UniGene Anatomical Profiling Dothiepin  Aliases 172130 18.000000 PubChem-Compound N/A 3H-QNB  Aliases HUMAN CLONED Stanton T, et al., 1993
 
42010 Cholinergic, muscarinic M2  Aliases NCBI - UniGene Anatomical Profiling Dothiepin  Aliases 172130 109.000000 PubChem-Compound N/A 3H-QNB  Aliases HUMAN CLONED Stanton T, et al., 1993
 
42029 Cholinergic, muscarinic M3  Aliases NCBI - UniGene Anatomical Profiling Dothiepin  Aliases 172130 38.000000 PubChem-Compound N/A 3H-QNB  Aliases HUMAN CLONED Stanton T, et al., 1993
 
42048 Cholinergic, muscarinic M4  Aliases NCBI - UniGene Anatomical Profiling Dothiepin  Aliases 172130 61.000000 PubChem-Compound N/A 3H-QNB  Aliases HUMAN CLONED Stanton T, et al., 1993
 
42067 Cholinergic, muscarinic M5  Aliases NCBI - UniGene Anatomical Profiling Dothiepin  Aliases 172130 92.000000 PubChem-Compound N/A 3H-QNB  Aliases HUMAN CLONED Stanton T, et al., 1993
 
37218 Dopamine Transporter  Aliases NCBI - UniGene N/A Dothiepin  Aliases 172130 5,185.000000 PubChem-Compound N/A 3H-DA UPTAKE  Aliases RAT STRIATUM Sanchez C, et al., 1999
 
45576 Dopamine Transporter  Aliases NCBI - UniGene N/A Dothiepin  Aliases 172130 5,310.000000 PubChem-Compound N/A 3H-WIN 35,428  Aliases HUMAN CLONED Tatsumi M, et al., 1997
 
37321 HISTAMINE H1  Aliases NCBI - UniGene Anatomical Profiling Dothiepin  Aliases 172130 4.000000 PubChem-Compound N/A 3H-MEPYRAMINE  Aliases RAT BRAIN Sanchez C, et al., 1999
 
37207 Norepinephrine transporter  Aliases N/A N/A Dothiepin  Aliases 172130 70.000000 PubChem-Compound N/A 3H-NE Uptake  Aliases RAT CORTEX Sanchez C, et al., 1999
 
45575 Norepinephrine transporter  Aliases N/A N/A Dothiepin  Aliases 172130 46.000000 PubChem-Compound N/A 3H-Nisoxetine  Aliases HUMAN CLONED Tatsumi M, et al., 1997
 


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