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The database has 60243Ki values for searching, and is growing
This list shows the Top 100 Receptors/Targets in Ki
Please let us know if you feel we should add any papers or data. We welcome all feedback/suggestions/comments
Other features on Ki DB are: Download Ki, Data Mining, CDD Interface allows mining Ki database by structure, substructure or structure similarity.
Anatomical profiling of GPCR expression is offered for selected targets.

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Your search returned 9 results:

IDReceptor/AliasesUniGeneAnat. ProfilingTest Ligand Name/AliasesNCIKi (nM)PubChemChEMBLHot Ligand/AliasesSpeciesSourceReference
45640 5-HT Transporter  Aliases NCBI - UniGene N/A Protriptyline  Aliases N/A 19.600000 PubChem-Compound ChEMBL 3H-IMIPRAMINE  Aliases HUMAN CLONED Tatsumi M, et al., 1997
 
62813 Alpha 1 Adrenergic Receptor  Aliases N/A N/A Protriptyline  Aliases N/A 130.000000 PubChem-Compound ChEMBL 3H-PRAZOSIN  Aliases HUMAN Brain Frontal Cortex Richelson, Elliott et. al, 1984
 
62842 Alpha 2 Adrenergic Receptor  Aliases N/A N/A Protriptyline  Aliases N/A 6,600.000000 PubChem-Compound ChEMBL 3H-RAUWOLSCINE  Aliases HUMAN Brain Frontal Cortex Richelson, Elliott et. al, 1984
 
62865 D2  Aliases N/A N/A Protriptyline  Aliases N/A 2,300.000000 PubChem-Compound ChEMBL 3H-SPIROPERIDOL  Aliases HUMAN Brain caudate nucleus Richelson, Elliott et. al, 1984
 
45642 Dopamine Transporter  Aliases NCBI - UniGene N/A Protriptyline  Aliases N/A 2,100.000000 PubChem-Compound ChEMBL 3H-WIN 35,428  Aliases HUMAN CLONED Tatsumi M, et al., 1997
 
62760 H1  Aliases N/A N/A Protriptyline  Aliases N/A 25.000000 PubChem-Compound ChEMBL 3H-doxepin  Aliases HUMAN Brain Frontal Cortex Richelson, Elliott et. al, 1984
 
13055 HISTAMINE H1  Aliases NCBI - UniGene Anatomical Profiling Protriptyline  Aliases N/A 60.000000 PubChem-Compound ChEMBL 3H-MEPYRAMINE  Aliases RAT BRAIN Tran VT, et al., 1978
 
62776 Muscarinic Acetylcholine Receptor  Aliases N/A N/A Protriptyline  Aliases N/A 25.000000 PubChem-Compound ChEMBL 3H-QNB  Aliases HUMAN Brain caudate nucleus Richelson, Elliott et. al, 1984
 
45641 Norepinephrine transporter  Aliases N/A N/A Protriptyline  Aliases N/A 1.410000 PubChem-Compound ChEMBL 3H-Nisoxetine  Aliases HUMAN CLONED Tatsumi M, et al., 1997
 


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